Number

Class

Target

Targets (gene)

目标(基因)

Assay Format

Agonist Mode

Antagonist Mode

Price

1

GPCR

β1

β1-adrenergic receptor (ADRB1)

β1肾上腺素能受体

cAMP

+

+

1800

2

β2

β2-adrenergic receptor (ADRB2)

β2肾上腺素能受体

cAMP

+

+

1800

3

op-delta

δ-type opioid receptor (OPRD1)

δ型阿片受体

cAMP

+

+

1800

4

op-kappa

κ-type opioid receptor (OPRK1)

κ型阿片受体

cAMP

+

+

1800

5

op-mu

μ-type opioid receptor (OPRM1)

μ型阿片受体

cAMP

+

+

1800

6

Transporter

NET

Noradrenaline transporter (SLC6A2)

去甲肾上腺素转运蛋白(SLC6A2)

Uptake

－

+

1500

7

DAT

Dopamine transporter (SLC6A3)

多巴胺转运蛋白(SLC6A3)

Uptake

－

+

1500

Summary

12000